NEVÍDALOVÁ, Hana, Lenka MICHALCOVÁ a Zdeněk GLATZ. STUDYING OF COMPETITIVE INTERACTIONS OF DRUGS WITH HUMAN SERUM ALBUMIN BY CAPILLARY ELECTROPHORESIS-FRONTAL ANALYSIS. Online. In František Foret, Jana Křenková, Iveta Drobníková, Karel Klepárník. 13 th International Interdisciplinary Meeting on Bioanalysis CECE 2016. Brno, Czech Republic: Institute of Analytical Chemistry of the CAS, v. v. i., Brno, Czech Republic, 2016, s. 202-205. ISBN 978-80-904959-4-4. |
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@inproceedings{1363886, author = {Nevídalová, Hana and Michalcová, Lenka and Glatz, Zdeněk}, address = {Brno, Czech Republic}, booktitle = {13 th International Interdisciplinary Meeting on Bioanalysis CECE 2016}, editor = {František Foret, Jana Křenková, Iveta Drobníková, Karel Klepárník.}, keywords = {capillary electrophoresis-frontal analysis; competitive interaction; albumin}, howpublished = {elektronická verze "online"}, language = {eng}, location = {Brno, Czech Republic}, isbn = {978-80-904959-4-4}, pages = {202-205}, publisher = {Institute of Analytical Chemistry of the CAS, v. v. i., Brno, Czech Republic}, title = {STUDYING OF COMPETITIVE INTERACTIONS OF DRUGS WITH HUMAN SERUM ALBUMIN BY CAPILLARY ELECTROPHORESIS-FRONTAL ANALYSIS}, url = {http://www.ce-ce.org}, year = {2016} }
TY - JOUR ID - 1363886 AU - Nevídalová, Hana - Michalcová, Lenka - Glatz, Zdeněk PY - 2016 TI - STUDYING OF COMPETITIVE INTERACTIONS OF DRUGS WITH HUMAN SERUM ALBUMIN BY CAPILLARY ELECTROPHORESIS-FRONTAL ANALYSIS PB - Institute of Analytical Chemistry of the CAS, v. v. i., Brno, Czech Republic CY - Brno, Czech Republic SN - 9788090495944 KW - capillary electrophoresis-frontal analysis KW - competitive interaction KW - albumin UR - http://www.ce-ce.org N2 - Drug-protein interactions have a significant effect on pharmacodynamics and pharmacokinetics properties of drugs. Bound fraction of drugs is reservoir, whereas free fraction provides pharmacological effect.Study of drug-protein interactions is thus important in the clinical therapy and in the development of new drugs.In this study displacement of L tryptophan from its binding site on human serum albumin (HSA) by several drugs was investigated by capillary electrophoresis frontal analysis (CE-FA). ER -
NEVÍDALOVÁ, Hana, Lenka MICHALCOVÁ a Zdeněk GLATZ. STUDYING OF COMPETITIVE INTERACTIONS OF DRUGS WITH HUMAN SERUM ALBUMIN BY CAPILLARY ELECTROPHORESIS-FRONTAL ANALYSIS. Online. In František Foret, Jana Křenková, Iveta Drobníková, Karel Klepárník. \textit{13 th International Interdisciplinary Meeting on Bioanalysis CECE 2016}. Brno, Czech Republic: Institute of Analytical Chemistry of the CAS, v. v. i., Brno, Czech Republic, 2016, s.~202-205. ISBN~978-80-904959-4-4.
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