J 2021

Prehľad biorelevantných dynamických disolučných prístrojov

BÍLIK, Tomáš, Ivan STUPÁK, Jakub VYSLOUŽIL, Martin ČULEN, Jiří DOHNAL et. al.

Basic information

Original name

Prehľad biorelevantných dynamických disolučných prístrojov

Name (in English)

An Overview of Biorelevant Dynamic Dissolution Instruments

Authors

BÍLIK, Tomáš (203 Czech Republic, belonging to the institution), Ivan STUPÁK (703 Slovakia, guarantor, belonging to the institution), Jakub VYSLOUŽIL (203 Czech Republic, belonging to the institution), Martin ČULEN (703 Slovakia, belonging to the institution) and Jiří DOHNAL (203 Czech Republic, belonging to the institution)

Edition

CHEMICKÉ LISTY, Praha, Česká společnost chemická, 2021, 0009-2770

Other information

Language

Slovak

Type of outcome

Článek v odborném periodiku

Field of Study

30104 Pharmacology and pharmacy

Country of publisher

Czech Republic

Confidentiality degree

není předmětem státního či obchodního tajemství

References:

Impact factor

Impact factor: 0.356

RIV identification code

RIV/00216224:14160/21:00123928

Organization unit

Faculty of Pharmacy

UT WoS

000738342100005

Keywords in English

solid oral dosage forms; biorelevant dissolution test; in vitro gastrointestinal system

Tags

Tags

International impact, Reviewed
Změněno: 28/8/2024 11:36, Mgr. Michal Petr

Abstract

V originále

The use of solid oral dosage forms depends on the degree of bioavailability of the active pharmaceutical ingredient. The rate and extent of the drug released from the dosage form and subsequently dissolved in the gastrointestinal fluids greatly affects its fate in the human body. In vitro dissolution test may provide an in-depth understanding of a drug formulation's behaviour in vivo, as long as it sufficiently simulates relevant gastrointestinal conditions. Therefore, the development of in vitro gastrointestinal systems, which reflects advanced technology and knowledge about the human body, is receiving considerable attention. This article is focused on the biorelevant dynamic apparatuses and their sophisticated design, overcoming many limitations of conventional dissolution devices and allowing a better correlation with in vivo behaviour of solid oral dosage forms.

In English

The use of solid oral dosage forms depends on the degree of bioavailability of the active pharmaceutical ingredient. The rate and extent of the drug released from the dosage form and subsequently dissolved in the gastrointestinal fluids greatly affects its fate in the human body. In vitro dissolution test may provide an in-depth understanding of a drug formulation's behaviour in vivo, as long as it sufficiently simulates relevant gastrointestinal conditions. Therefore, the development of in vitro gastrointestinal systems, which reflects advanced technology and knowledge about the human body, is receiving considerable attention. This article is focused on the biorelevant dynamic apparatuses and their sophisticated design, overcoming many limitations of conventional dissolution devices and allowing a better correlation with in vivo behaviour of solid oral dosage forms.