DOSTÁLEK, Miroslav, Veronika MINAŘÍKOVÁ, Jan JUŘICA, Josef TOMANDL a Eva HADAŠOVÁ. Methamphetamine increases CYP2D1/2 activity in isolated perfused rat liver. Psychiatrie. Praha: Tigis, 2004, roč. 8, Suppl. 4, s. 19-19. ISSN 1211-7579. |
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@article{563276, author = {Dostálek, Miroslav and Minaříková, Veronika and Juřica, Jan and Tomandl, Josef and Hadašová, Eva}, article_location = {Praha}, article_number = {Suppl. 4}, keywords = {methamphetamine; rat; liver}, language = {cze}, issn = {1211-7579}, journal = {Psychiatrie}, title = {Methamphetamine increases CYP2D1/2 activity in isolated perfused rat liver}, volume = {8}, year = {2004} }
TY - JOUR ID - 563276 AU - Dostálek, Miroslav - Minaříková, Veronika - Juřica, Jan - Tomandl, Josef - Hadašová, Eva PY - 2004 TI - Methamphetamine increases CYP2D1/2 activity in isolated perfused rat liver JF - Psychiatrie VL - 8 IS - Suppl. 4 SP - 19-19 EP - 19-19 PB - Tigis SN - 12117579 KW - methamphetamine KW - rat KW - liver N2 - Methamphetamine represents a significant drug abuse problem in many European countries including the Czech republic. Studies in human liver microsomes have shown that crucial metabolic reactions of MeAmp are catalyzed by CYP2D6; furthermore, some amphetamine analogues were reported as inhibitors of CYP2D6 (Wu et. al., 1997). The aim of the study was to ascertain the influence of acute and repeated pretreatment of rats with various doses of methamphetamine on metabolic activity of CYP2D1/2 (correlate of human CYP2D6) in the isolated perfused rat liver. ER -
DOSTÁLEK, Miroslav, Veronika MINAŘÍKOVÁ, Jan JUŘICA, Josef TOMANDL a Eva HADAŠOVÁ. Methamphetamine increases CYP2D1/2 activity in isolated perfused rat liver. \textit{Psychiatrie}. Praha: Tigis, 2004, roč.~8, Suppl. 4, s.~19-19. ISSN~1211-7579.
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