BÉBAROVÁ, Markéta, Peter MATEJOVIČ, Michal PÁSEK and Marie NOVÁKOVÁ. Effect of haloperidol on transient outward potassium current in rat ventricular myocytes. European Journal of Pharmacology. Amsterdam, The Netherlands: Elsevier Science B.V., 2006, vol. 550, 1-3, p. 15-23. ISSN 0014-2999. |
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@article{700534, author = {Bébarová, Markéta and Matejovič, Peter and Pásek, Michal and Nováková, Marie}, article_location = {Amsterdam, The Netherlands}, article_number = {1-3}, keywords = {haloperidol; transient outward current; sigma receptors; rat ventricular myocytes; whole-cell pach clamp; quantitative model}, language = {eng}, issn = {0014-2999}, journal = {European Journal of Pharmacology}, title = {Effect of haloperidol on transient outward potassium current in rat ventricular myocytes}, volume = {550}, year = {2006} }
TY - JOUR ID - 700534 AU - Bébarová, Markéta - Matejovič, Peter - Pásek, Michal - Nováková, Marie PY - 2006 TI - Effect of haloperidol on transient outward potassium current in rat ventricular myocytes JF - European Journal of Pharmacology VL - 550 IS - 1-3 SP - 15-23 EP - 15-23 PB - Elsevier Science B.V. SN - 00142999 KW - haloperidol KW - transient outward current KW - sigma receptors KW - rat ventricular myocytes KW - whole-cell pach clamp KW - quantitative model N2 - Haloperidol induced a decrease of amplitude and an acceleration of apparent inactivation of transient outward potassium current (Ito), both in a voltage-dependent manner. The averaged inhibition of Ito, evaluated as a change of its time integral, was 23.0 +/- 3.2% at stimulation frequency of 0.1 Hz. As a consequence of slow recovery of Ito from the haloperidol-induced block (time constant 1482 +/- 83 ms), a cumulation of the block up to about 40% appeared at 3.3 Hz. ER -
BÉBAROVÁ, Markéta, Peter MATEJOVIČ, Michal PÁSEK and Marie NOVÁKOVÁ. Effect of haloperidol on transient outward potassium current in rat ventricular myocytes. \textit{European Journal of Pharmacology}. Amsterdam, The Netherlands: Elsevier Science B.V., 2006, vol.~550, 1-3, p.~15-23. ISSN~0014-2999.
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