NEVÍDALOVÁ, Hana, Lenka MICHALCOVÁ a Zdeněk GLATZ. Applicability of capillary electrophoresis-frontal analysis for displacement studies: effect of several drugs on L-tryptophan and lidocaine binding to human serum albumin. Journa of Separation Science. Weinheim: Wiley-VCH, 2020, roč. 43, č. 22, s. 4225-4233. ISSN 1615-9306. Dostupné z: https://dx.doi.org/10.1002/jssc.202000594. |
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@article{1679993, author = {Nevídalová, Hana and Michalcová, Lenka and Glatz, Zdeněk}, article_location = {Weinheim}, article_number = {22}, doi = {http://dx.doi.org/10.1002/jssc.202000594}, keywords = {CE; Albumin; Drug}, language = {eng}, issn = {1615-9306}, journal = {Journa of Separation Science}, title = {Applicability of capillary electrophoresis-frontal analysis for displacement studies: effect of several drugs on L-tryptophan and lidocaine binding to human serum albumin}, url = {https://doi.org/10.1002/jssc.202000594}, volume = {43}, year = {2020} }
TY - JOUR ID - 1679993 AU - Nevídalová, Hana - Michalcová, Lenka - Glatz, Zdeněk PY - 2020 TI - Applicability of capillary electrophoresis-frontal analysis for displacement studies: effect of several drugs on L-tryptophan and lidocaine binding to human serum albumin JF - Journa of Separation Science VL - 43 IS - 22 SP - 4225-4233 EP - 4225-4233 PB - Wiley-VCH SN - 16159306 KW - CE KW - Albumin KW - Drug UR - https://doi.org/10.1002/jssc.202000594 L2 - https://doi.org/10.1002/jssc.202000594 N2 - In this study, the binding characteristics of six drugs with human serum albumin, the most abundant protein in human plasma, were determined by capillary electrophoresis-frontal analysis, and the obtained values of binding parameters were compared with the literature data. The affect of several drugs and site markers on the binding of L-tryptophan and lidocaine to human serum albumin was investigated in subsequent displacement studies which thus demonstrated the usability of capillary electrophoresis as an automated high-throughput screening method for drug-protein binding studies. ER -
NEVÍDALOVÁ, Hana, Lenka MICHALCOVÁ a Zdeněk GLATZ. Applicability of capillary electrophoresis-frontal analysis for displacement studies: effect of several drugs on L-tryptophan and lidocaine binding to human serum albumin. \textit{Journa of Separation Science}. Weinheim: Wiley-VCH, 2020, roč.~43, č.~22, s.~4225-4233. ISSN~1615-9306. Dostupné z: https://dx.doi.org/10.1002/jssc.202000594.
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