CHRISTÉ, Georg, Habiba TEBBAKH, Milena ŠIMURDOVÁ, Rémi FORRAT a Jiří ŠIMURDA. Propafenone blocks ATP-sensitive K+ channels in rabbit atrial and ventricular cardiomyocytes. European Journal of Pharmacology. Amsterdam: Elsevier Science B.V., 1999, roč. 373, 2-3, s. 223-232. ISSN 0014-2999. |
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@article{219531, author = {Christé, Georg and Tebbakh, Habiba and Šimurdová, Milena and Forrat, Rémi and Šimurda, Jiří}, article_location = {Amsterdam}, article_number = {2-3}, keywords = {Antiarrhythmic; Propafenone; K+ channel; ATP-sensitive; Cardiomyocyte; Ventricle.}, language = {eng}, issn = {0014-2999}, journal = {European Journal of Pharmacology}, title = {Propafenone blocks ATP-sensitive K+ channels in rabbit atrial and ventricular cardiomyocytes.}, volume = {373}, year = {1999} }
TY - JOUR ID - 219531 AU - Christé, Georg - Tebbakh, Habiba - Šimurdová, Milena - Forrat, Rémi - Šimurda, Jiří PY - 1999 TI - Propafenone blocks ATP-sensitive K+ channels in rabbit atrial and ventricular cardiomyocytes. JF - European Journal of Pharmacology VL - 373 IS - 2-3 SP - 223 EP - 223 PB - Elsevier Science B.V. SN - 00142999 KW - Antiarrhythmic KW - Propafenone KW - K+ channel KW - ATP-sensitive KW - Cardiomyocyte KW - Ventricle. N2 - Propafenone, a class I antiarrhythmic agent, inhibits several membrane currents, however, its effect on ATP-sensitive potassium current (IKATP) of cerdiac cells have not been tested. We evaluated the blocking effect of 0.1 to 100 uM propafenone on the whole cell IKATP as triggered by dinitrophenol in aduld rabbit isolated atrial and ventricular cardiomyocytes. It is concluded that propafenone blocks cardiac IKATP at a single site. This block might play a role in the beneficial and adverse effects of the drug. ER -
CHRISTÉ, Georg, Habiba TEBBAKH, Milena ŠIMURDOVÁ, Rémi FORRAT a Jiří ŠIMURDA. Propafenone blocks ATP-sensitive K+ channels in rabbit atrial and ventricular cardiomyocytes. \textit{European Journal of Pharmacology}. Amsterdam: Elsevier Science B.V., 1999, roč.~373, 2-3, s.~223-232. ISSN~0014-2999.
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