D 2009

Benzoin as a photoremovable chiral auxiliary

KAMMATH, Viju Balachandran; Peter ŠEBEJ; Tomáš SLANINA a Petr KLÁN

Základní údaje

Originální název

Benzoin as a photoremovable chiral auxiliary

Název česky

Benzoin jako fotolabilní chirální induktor

Autoři

KAMMATH, Viju Balachandran; Peter ŠEBEJ; Tomáš SLANINA a Petr KLÁN

Vydání

Washington, USA, 238th American Chemical Society National Meeting & Exposition, 1 s. 2009

Nakladatel

American Chemical Society

Další údaje

Jazyk

angličtina

Typ výsledku

Stať ve sborníku

Obor

10401 Organic chemistry

Stát vydavatele

Spojené státy

Utajení

není předmětem státního či obchodního tajemství

Označené pro přenos do RIV

Ne

Organizační jednotka

Přírodovědecká fakulta

ISBN

978-0-8412-0005-0

Klíčová slova česky

Benzoin; Chirální Induktor; Fotochemie; Fotolabilní skupina; Diels-Aderova reakce

Klíčová slova anglicky

Benzoin; Chiral Auxiliary; Photochemistry; Photoremovable Protecting Group; Diels-Alder Reaction

Příznaky

Mezinárodní význam
Změněno: 26. 3. 2010 13:32, Mgr. Peter Šebej, Ph.D.

Anotace

V originále

Controlling the reaction stereochemistry is often achieved by using a chiral auxiliary which is covalently attached to the prochiral substrate before chirality relay is performed. These groups are optically active compounds or units that are temporarily incorporated to be utilized in the selective formation of one of the enantiomers. Here photoremovable chiral auxiliary (PCA) represents a new strategy in the field of asymmetric organic synthesis, which offers a chiral auxiliary that can be photochemically removed under specific conditions. The benzoin group is known to be a good photoremovable protecting group for a variety of functionalities, such as carboxylates, hydroxyls, phosphates etc. Since benzoin contains a chiral center, we proposed and studied its derivatives as PCA. Enantiopure benzoin group is connected to a dienophile which reacts with a diene in the presence of various catalysts. The auxiliary is then removed upon irradiation giving the products exhibiting enantiomeric excess.

Česky

Controlling the reaction stereochemistry is often achieved by using a chiral auxiliary which is covalently attached to the prochiral substrate before chirality relay is performed. These groups are optically active compounds or units that are temporarily incorporated to be utilized in the selective formation of one of the enantiomers. Here photoremovable chiral auxiliary (PCA) represents a new strategy in the field of asymmetric organic synthesis, which offers a chiral auxiliary that can be photochemically removed under specific conditions. The benzoin group is known to be a good photoremovable protecting group for a variety of functionalities, such as carboxylates, hydroxyls, phosphates etc. Since benzoin contains a chiral center, we proposed and studied its derivatives as PCA. Enantiopure benzoin group is connected to a dienophile which reacts with a diene in the presence of various catalysts. The auxiliary is then removed upon irradiation giving the products exhibiting enantiomeric excess.

Návaznosti

ME09021, projekt VaV
Název: Vývoj nových fotoaktivovatelných systémů pro biologické studie
Investor: Ministerstvo školství, mládeže a tělovýchovy ČR, Vývoj nových fotoaktivovatelných systémů pro biologické studie, Program výzkumu a vývoje KONTAKT (ME)