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@inproceedings{563064, author = {Juřica, Jan and Dostálek, Miroslav and Tomandl, Josef and Hadašová, Eva}, address = {Olomouc}, booktitle = {ACTA UNIVERISTATIS PALACKIANAE OLOMUCENSIS FACULTAS RERUM NATURALIUM}, keywords = {Midazolam; CYP-450}, language = {cze}, location = {Olomouc}, isbn = {80-244-0882-1}, pages = {218-218}, publisher = {Univerzita Palackého Olomouc}, title = {Determination of Midazolam from Perfuse Medium as a Probe Substrate of Cytochrome P450 3A1/2 Activity in Rats}, year = {2004} }
TY - JOUR ID - 563064 AU - Juřica, Jan - Dostálek, Miroslav - Tomandl, Josef - Hadašová, Eva PY - 2004 TI - Determination of Midazolam from Perfuse Medium as a Probe Substrate of Cytochrome P450 3A1/2 Activity in Rats PB - Univerzita Palackého Olomouc CY - Olomouc SN - 8024408821 KW - Midazolam KW - CYP-450 N2 - The aim of the project was to develop HPLC method for determination of midazolam and its three metabolites, 1- and 4-hydroxymidazolam and 1,4-dihydroxymidazolam from perfuse rat liver medium. Hydroxylation of midazolam is used as a valuable tool for measurement of metabolic activity of the 3A1/2 isoform of cytochrome P-450 in rats (CYP3A1/2)This method is simple, rapid, sensitive and applicable for modeling and description of possible pharmacological interactions on rat CYP3A1/2. ER -
JUŘICA, Jan, Miroslav DOSTÁLEK, Josef TOMANDL a Eva HADAŠOVÁ. Determination of Midazolam from Perfuse Medium as a Probe Substrate of Cytochrome P450 3A1/2 Activity in Rats. In \textit{ACTA UNIVERISTATIS PALACKIANAE OLOMUCENSIS FACULTAS RERUM NATURALIUM}. Olomouc: Univerzita Palackého Olomouc, 2004, s.~218-218. ISBN~80-244-0882-1.
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