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Convergent Assembly of the Tricyclic Labdane Core Enables Synthesis of Diverse Forskolin-like Molecules J - Článek v odborném periodikuSZCZEPANIK, Pawel Marcin; Andrey MIKHAYLOV; Ondřej HYLSE; Roman KUČERA; Petra DAĎOVÁ; Marek NEČAS; Lukáš KUBALA; Kamil PARUCH a Jakub ŠVENDA. Convergent Assembly of the Tricyclic Labdane Core Enables Synthesis of Diverse Forskolin-like Molecules. Angewandte Chemie International Edition. Wiley, 2023, roč. 62, č. 1, s. 1-7. ISSN 1433-7851. Dostupné z: https://doi.org/10.1002/anie.202213183.Podrobněji: https://is.muni.cz/publication/2249874/cs
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A Concise Synthesis of Forskolin J - Článek v odborném periodikuHYLSE, Ondřej; Lukáš MAIER; Roman KUČERA; Tomáš PEREČKO; Aneta SVOBODOVÁ; Lukáš KUBALA; Kamil PARUCH a Jakub ŠVENDA. A Concise Synthesis of Forskolin. Angewandte Chemie International Edition. Německo: Verlag Chemie, 2017, roč. 2017, č. 56, s. 12586-12589. ISSN 1433-7851. Dostupné z: https://doi.org/10.1002/anie.201706809.Podrobněji: https://is.muni.cz/publication/1392287/cs
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BRCA1 or CDK12 loss sensitizes cells to CHK1 inhibitors J - Článek v odborném periodikuPACULOVÁ, Hana; Juraj KRAMARA; Šárka ŠIMEČKOVÁ; Radek FEDR; Karel SOUČEK; Ondřej HYLSE; Kamil PARUCH; Marek SVOBODA; Martin MISTRÍK a Jiří KOHOUTEK. BRCA1 or CDK12 loss sensitizes cells to CHK1 inhibitors. Tumor Biology. Springer Netherlands, 2017, roč. 2017, October, s. 1-11. ISSN 1010-4283. Dostupné z: https://doi.org/10.1177/1010428317727479.Podrobněji: https://is.muni.cz/publication/1392816/cs
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Diastereoselective Flexible Synthesis of Carbocyclic C Nucleosides J - Článek v odborném periodikuMAIER, Lukáš; PrashantKumar KHIRSARIYA; Ondřej HYLSE; Santosh Kumar ADLA; Lenka ČERNOVÁ; Michal POLJAK; Soňa KRAJČOVIČOVÁ; Erik WEIS; Stanislav DRÁPELA; Karel SOUČEK a Kamil PARUCH. Diastereoselective Flexible Synthesis of Carbocyclic C Nucleosides. The Journal of Organic Chemistry. WASHINGTON, DC USA: American Chemical Society, 2017, roč. 82, č. 7, s. 3382-3402. ISSN 0022-3263. Dostupné z: https://doi.org/10.1021/acs.joc.6b02594.Podrobněji: https://is.muni.cz/publication/1382487/cs
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Synthesis and Profiling of a Novel Potent Selective Inhibitor of CHK1 Kinase Possessing Unusual N-trifluoromethylpyrazole Pharmacophore Resistant to Metabolic N-dealkylation J - Článek v odborném periodikuSAMADDER, Pounami; Tereza SUCHÁNKOVÁ; Ondřej HYLSE; PrashantKumar KHIRSARIYA; Fedor NIKULENKOV; Stanislav DRÁPELA; Nicol STRAKOVÁ; Petr VAŇHARA; Kateřina VAŠÍČKOVÁ; Hana KOLÁŘOVÁ; Lucia BINÓ; Miroslava BITTOVÁ; Petra OVESNÁ; Peter KOLLÁR; Radek FEDR; Milan EŠNER; Josef JAROŠ; Aleš HAMPL; Lumír KREJČÍ; Kamil PARUCH a Karel SOUČEK. Synthesis and Profiling of a Novel Potent Selective Inhibitor of CHK1 Kinase Possessing Unusual N-trifluoromethylpyrazole Pharmacophore Resistant to Metabolic N-dealkylation. Molecular Cancer Therapeutics. Philadelphia: American Association for Cancer Research, 2017, roč. 16, č. 9, s. 1831-1842. ISSN 1535-7163. Dostupné z: https://doi.org/10.1158/1535-7163.MCT-17-0018.Podrobněji: https://is.muni.cz/publication/1388764/cs
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Development and validation of a highly sensitive LC-MS method for determination of checkpoint kinase 1 inhibitors in mouse plasma D - Stať ve sborníkuBITTOVÁ, Miroslava; Hana KOLÁŘOVÁ; Ondřej HYLSE; PrashantKumar KHIRSARIYA a Kamil PARUCH. Development and validation of a highly sensitive LC-MS method for determination of checkpoint kinase 1 inhibitors in mouse plasma. In Vítězslav Maier. Advances in chromatography and electrophoresis & Chiranal 2016. Olomouc: Palacký University, Olomouc, 2016, s. 79-80. ISBN 978-80-244-4961-6.Podrobněji: https://is.muni.cz/publication/1347658/cs
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Checkpoint kinase 1 inhibition potentiates apoptosis and inflicts mitotic failure in CLL-derived MEC-1 cell line. a - Konferenční abstraktZEMANOVÁ, Jana; Ondřej HYLSE; Jana ČOLLÁKOVÁ; Petr VESELÝ; Alexandra OLTOVÁ; Kamil PARUCH a Martin TRBUŠEK. Checkpoint kinase 1 inhibition potentiates apoptosis and inflicts mitotic failure in CLL-derived MEC-1 cell line. In Haematologica (2016); 101(s1): 425. (21st Congress of the EHA). 2016.Podrobněji: https://is.muni.cz/publication/1363957/cs
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Chk1 inhibition significantly potentiates activity of nucleoside analogs in TP53-mutated B-lymphoid cells J - Článek v odborném periodikuZEMANOVÁ, Jana; Ondřej HYLSE; Jana COLLAKOVA; Pavel VESELY; Alexandra OLTOVÁ; Marek BORSKÝ; Kristína ZÁPRAŽNÁ; Marie KAŠPÁRKOVÁ; Pavlína JANOVSKÁ; Jan VERNER; Jiri KOHOUTEK; Marta DZIMKOVA; Vítězslav BRYJA; Zuzana JAŠKOVÁ; Yvona BRYCHTOVÁ; Kamil PARUCH a Martin TRBUŠEK. Chk1 inhibition significantly potentiates activity of nucleoside analogs in TP53-mutated B-lymphoid cells. Oncotarget. Albany: Impact Journals, 2016, roč. 7, č. 38, s. 62091-62106. ISSN 1949-2553. Dostupné z: https://doi.org/10.18632/oncotarget.11388.Podrobněji: https://is.muni.cz/publication/1363771/cs
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Facile rearrangements of a vinylogous alpha-hydroxy-beta-dicarbonyl substrate involving an apparent oxirane C-C bond scission J - Článek v odborném periodikuKUČERA, Roman; Ondřej HYLSE; Michal BABIAK a Jakub ŠVENDA. Facile rearrangements of a vinylogous alpha-hydroxy-beta-dicarbonyl substrate involving an apparent oxirane C-C bond scission. Tetrahedron Letters. OXFORD: Pergamon Press, 2015, roč. 56, č. 45, s. 6171-6173. ISSN 0040-4039. Dostupné z: https://doi.org/10.1016/j.tetlet.2015.09.015.Podrobněji: https://is.muni.cz/publication/1375990/cs
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Chronic lymphocytic leukemia cells are highly susceptible to direct inhibition of checkpoint kinase a - Konferenční abstraktZEMANOVÁ, Jana; Kamil PARUCH; Lumír KREJČÍ; Karel SOUČEK; Ondřej HYLSE; Miroslav BOUDNÝ; Marek BORSKÝ; Jitka OSIČKOVÁ; PrashantKumar KHIRSARIYA; Ludmila ŠEBEJOVÁ; Veronika NAVRKALOVÁ; Jitka MALČÍKOVÁ; Eva DIVÍŠKOVÁ; Yvona BRYCHTOVÁ; Jiří MAYER a Martin TRBUŠEK. Chronic lymphocytic leukemia cells are highly susceptible to direct inhibition of checkpoint kinase. In 20th Congress of the European Hematology Association in Haematologica. 2015.Podrobněji: https://is.muni.cz/publication/1315740/cs
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Exploring synthetic lethal interaction between Checkpoint Kinase 1(CHK1) and DNA replication stress k - Prezentace na konferencíchSAMADDER, Pounami. Exploring synthetic lethal interaction between Checkpoint Kinase 1(CHK1) and DNA replication stress. In HYLSE, Ondřej; Fedor NIKULENKOV; Tereza SUCHÁNKOVÁ; Karel SOUČEK; Kamil PARUCH a Lumír KREJČÍ. Cell Proliferation and Genome Integrity International symposium. 2014.Podrobněji: https://is.muni.cz/publication/1198372/cs
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Is checkpoint kinase 1 a suitable molecular target for combination with cancer chemotherapeutics? a - Konferenční abstraktZEMANOVÁ, Jana; Ludmila ŠEBEJOVÁ; Ondřej HYLSE; Kamil PARUCH; Šárka POSPÍŠILOVÁ a Martin TRBUŠEK. Is checkpoint kinase 1 a suitable molecular target for combination with cancer chemotherapeutics? In XXI. Biologické dny, Brno. 2014.Podrobněji: https://is.muni.cz/publication/1226598/cs
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Is checkpoint kinase 1 a suitable molecular target for sensitization of TP53-mutated leukemia and lymphoma cells to chemotherapy? a - Konferenční abstraktZEMANOVÁ, Jana; Ludmila ŠEBEJOVÁ; Ondřej HYLSE; Kamil PARUCH; Šárka POSPÍŠILOVÁ a Martin TRBUŠEK. Is checkpoint kinase 1 a suitable molecular target for sensitization of TP53-mutated leukemia and lymphoma cells to chemotherapy? In 16th International p53 workshop, Švédsko. 2014.Podrobněji: https://is.muni.cz/publication/1226646/cs
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New carbocyclic nucleosides: synthesis of carbocyclic pseudoisocytidine and its analogs J - Článek v odborném periodikuMAIER, Lukáš; Ondřej HYLSE; Marek NEČAS; Martin TRBUŠEK; Mari YTRE-ARNE; Bjorn DALHUS; Magnar BJORAS a Kamil PARUCH. New carbocyclic nucleosides: synthesis of carbocyclic pseudoisocytidine and its analogs. Tetrahedron Letters. 2014, roč. 55, č. 27, s. 3713-3716. ISSN 0040-4039. Dostupné z: https://doi.org/10.1016/j.tetlet.2014.05.030.Podrobněji: https://is.muni.cz/publication/1185536/cs
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Synthetic lethality in p53 mutated B-cell mylignancies: Chk-1 inhibition and DNA-PK inhibition effect in cell lines and primary CLL cells a - Konferenční abstraktZEMANOVÁ, Jana; Ludmila ŠEBEJOVÁ; Kamil PARUCH; Ondřej HYLSE; Šárka POSPÍŠILOVÁ; Jiří MAYER a Martin TRBUŠEK. Synthetic lethality in p53 mutated B-cell mylignancies: Chk-1 inhibition and DNA-PK inhibition effect in cell lines and primary CLL cells. In 18th Congress of the European Hematology Association in Haematologica, the hematology journal, Stockholm, Švédsko. 2013.Podrobněji: https://is.muni.cz/publication/1114363/cs
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Inhibice kinázy Chk1 senzitivuje buňky leukemií a lymfomů s mutacemi p53 na chemoterapeutika a - Konferenční abstraktZEMANOVÁ, Jana; Ludmila ŠEBEJOVÁ; Ondřej HYLSE; Kamil PARUCH; Šárka POSPÍŠILOVÁ a Martin TRBUŠEK. Inhibice kinázy Chk1 senzitivuje buňky leukemií a lymfomů s mutacemi p53 na chemoterapeutika. In XXVI. Olomoucké hematologické dny s mezinárodní účastí, Olomouc. 2012.Podrobněji: https://is.muni.cz/publication/1068297/cs
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Inhibition of Chk1 kinase sensitizes leukemia and lymphoma cell lines with TP53 mutations to chemotherapy a - Konferenční abstraktZEMANOVÁ, Jana; Ludmila ŠEBEJOVÁ; Ondřej HYLSE; Kamil PARUCH; Šárka PAVLOVÁ; Jiří MAYER; Šárka POSPÍŠILOVÁ a Martin TRBUŠEK. Inhibition of Chk1 kinase sensitizes leukemia and lymphoma cell lines with TP53 mutations to chemotherapy. In 54th ASH Annual Meeting and Exposition, Atlanta, USA in Blood. 2012.Podrobněji: https://is.muni.cz/publication/1083007/cs