Masarykova univerzita

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Filtrování publikací

    2023

    1. NĚMEC, Václav, PrashantKumar KHIRSARIYA, Pavlína JANOVSKÁ, Paula MARTÍN MOYANO, Lukáš MAIER, Petra PROCHÁZKOVÁ, Pavlína KEBKOVÁ, Tomáš GYBEĽ, Benedict-Tilman BERGER, Apirat CHAIKUAD, Maria REINECKE, Bernhard KUSTER, Stefan KNAPP, Vítězslav BRYJA a Kamil PARUCH. Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity. Angewandte Chemie International Edition. Wiley-VCH GmbH, 2023, roč. 62, č. 11, s. 1-7. ISSN 1433-7851. Dostupné z: https://dx.doi.org/10.1002/anie.202217532.

    2022

    1. ATTULURI, Venkata Pardha S., Juan Francisco SANCHEZ LOPEZ, Lukáš MAIER, Kamil PARUCH a Helene ROBERT BOISIVON. Comparing the efficiency of six clearing methods in developing seeds of Arabidopsis thaliana. Plant Reproduction. Springer, 2022, roč. 35, č. 4, s. 279-293. ISSN 2194-7953. Dostupné z: https://dx.doi.org/10.1007/s00497-022-00453-4.
    2. KHIRSARIYA, PrashantKumar, Patrik POSPÍŠIL, Lukáš MAIER, Miroslav BOUDNÝ, Martin BABÁŠ, Ondřej KROUTIL, Marek MRÁZ, Robert VÁCHA a Kamil PARUCH. Synthesis and Profiling of Highly Selective Inhibitors of Methyltransferase DOT1L Based on Carbocyclic C-Nucleosides. Journal of Medicinal Chemistry. Washington: American Chemical Society, 2022, roč. 65, č. 7, s. 5701-5723. ISSN 0022-2623. Dostupné z: https://dx.doi.org/10.1021/acs.jmedchem.1c02228.

    2021

    1. NĚMEC, Václav, Lukáš MAIER, Benedict-Tilman BERGER, Apirat CHAIKUAD, Stanislav DRÁPELA, Karel SOUČEK, Stefan KNAPP a Kamil PARUCH. Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core. European Journal of Medicinal Chemistry. Elsevier Masson s.r.l., 2021, roč. 215, April, s. "113299", 8 s. ISSN 0223-5234. Dostupné z: https://dx.doi.org/10.1016/j.ejmech.2021.113299.

    2019

    1. NĚMEC, Václav, Michaela HYLSOVÁ, Lukáš MAIER, Jana FLEGEL, Sonja SIEVERS, Slava ZIEGLER, Martin SCHRÖDER, Benedict-Tilman BERGER, Apirat CHAIKUAD, Barbora VALČÍKOVÁ, Stjepan ULDRIJAN, Stanislav DRÁPELA, Karel SOUČEK, Hebert WALDMANN, Stefan KNAPP a Kamil PARUCH. Furo[3,2-b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway. Angewandte Chemie International Edition. Weinheim: Wiley-VCH, 2019, roč. 58, č. 4, s. 1062-1066. ISSN 1433-7851. Dostupné z: https://dx.doi.org/10.1002/anie.201810312.

    2017

    1. HYLSE, Ondřej, Lukáš MAIER, Roman KUČERA, Tomáš PEREČKO, Aneta SVOBODOVÁ, Lukáš KUBALA, Kamil PARUCH a Jakub ŠVENDA. A Concise Synthesis of Forskolin. Angewandte Chemie International Edition. Německo: Verlag Chemie, 2017, roč. 2017, č. 56, s. 12586-12589. ISSN 1433-7851. Dostupné z: https://dx.doi.org/10.1002/anie.201706809.
    2. MAIER, Lukáš, PrashantKumar KHIRSARIYA, Ondřej HYLSE, Santosh Kumar ADLA, Lenka ČERNOVÁ, Michal POLJAK, Soňa KRAJČOVIČOVÁ, Erik WEIS, Stanislav DRÁPELA, Karel SOUČEK a Kamil PARUCH. Diastereoselective Flexible Synthesis of Carbocyclic C Nucleosides. The Journal of Organic Chemistry. WASHINGTON, DC USA: American Chemical Society, 2017, roč. 82, č. 7, s. 3382-3402. ISSN 0022-3263. Dostupné z: https://dx.doi.org/10.1021/acs.joc.6b02594.

    2015

    1. KOVÁČOVÁ, Silvia, Santosh Kumar ADLA, Lukáš MAIER, Michal BABIAK, Yoshiyuki MIZUSHINA a Kamil PARUCH. Synthesis of carbocyclic analogs of dehydroaltenusin: identification of a stable inhibitor of calf DNA polymerase a. Tetrahedron. Pergamon Press, 2015, roč. 71, č. 40, s. 7575-7582. ISSN 0040-4020. Dostupné z: https://dx.doi.org/10.1016/j.tet.2015.08.005.

    2014

    1. MAIER, Lukáš, Ondřej HYLSE, Marek NEČAS, Martin TRBUŠEK, Mari YTRE-ARNE, Bjorn DALHUS, Magnar BJORAS a Kamil PARUCH. New carbocyclic nucleosides: synthesis of carbocyclic pseudoisocytidine and its analogs. Tetrahedron Letters. 2014, roč. 55, č. 27, s. 3713-3716. ISSN 0040-4039. Dostupné z: https://dx.doi.org/10.1016/j.tetlet.2014.05.030.

    2013

    1. AMARO, Mariana, Jan BREZOVSKÝ, Silvia KOVÁČOVÁ, Lukáš MAIER, Radka CHALOUPKOVÁ, Jan SYKORA, Kamil PARUCH, Jiří DAMBORSKÝ a Martin HOF. Are Time-Dependent Fluorescence Shifts at the Tunnel Mouth of Haloalkane Dehalogenase Enzymes Dependent on the Choice of the Chromophore? Journal of Physical Chemistry B. WASHINGTON: AMER CHEMICAL SOC, 2013, roč. 117, č. 26, s. 7898-7906. ISSN 1520-6106. Dostupné z: https://dx.doi.org/10.1021/jp403708c.
    2. KADAM, Shivaji Sambhaji, Lukáš MAIER, Tomáš ŠOLOMEK, Marek NEČAS, Karel ŠMEJKAL, Jiří DOSTÁL, Vladimír SKLENÁŘ a Radek MAREK. Structure and NMR properties of 6-substituted-5,6-dihydrobenzo[c]phenanthridine alkaloids. Journal of Physical Organic Chemistry. Wiley, 2013, roč. 26, č. 10, s. 814-821. ISSN 0894-3230. Dostupné z: https://dx.doi.org/10.1002/poc.3175.
    3. KADAM, Shivaji Sambhaji, Lukáš MAIER, Ioannis KOSTAKIS, Nicole POULI, Jaromír TOUŠEK, Marek NEČAS, Panagiotis MARAKOS a Radek MAREK. Synthesis and Tautomerism of Substituted Pyrazolo[4,3-c]pyrazoles. European Journal of Organic Chemistry. Weinheim: WILEY-VCH, 2013, roč. 2013, č. 30, s. 6811-6822. ISSN 1434-193X. Dostupné z: https://dx.doi.org/10.1002/ejoc.201300606.

    2012

    1. KADAM, Shivaji Sambhaji, Jaromír TOUŠEK, Lukáš MAIER, Matej PIPÍŠKA, Vladimír SKLENÁŘ a Radek MAREK. Understanding the NMR properties and conformational behavior of indole vs. azaindole group in protoberberines: NICS and NCS analysis. Journal of Molecular Structure. Amsterdam: Elsevier, 2012, roč. 1028, Nov, s. 31-38. ISSN 0022-2860. Dostupné z: https://dx.doi.org/10.1016/j.molstruc.2012.06.034.

    2010

    1. MAIER, Lukáš, Tomáš ŠOLOMEK, Matej PIPÍŠKA, Zdeněk KŘÍŽ, Marek NEČAS a Radek MAREK. Structural study of 8-azole derivatives of protoberberine alkaloids: experimental and quantum chemical approach. Tetrahedron. Oxford, England: Pergamon - Elsevier Science, 2010, roč. 66, č. 47, s. 9277-9285. ISSN 0040-4020.

    2008

    1. GRYCOVÁ, Lenka, Dagmar HULOVÁ, Lukáš MAIER, Stanislav STANDARA, Marek NEČAS, Filip LEMIÉRE, Radovan KAREŠ, Jiří DOSTÁL a Radek MAREK. Covalent bonding of azoles to quaternary protoberberine alkaloids. Magnetic Resonance in Chemistry. John Wiley & Sons, 2008, roč. 46, č. 12, s. 1127-1134. ISSN 0749-1581. Dostupné z: https://dx.doi.org/10.1002/mrc.2325.
    2. GRYCOVÁ, Lenka, Dagmar HULOVÁ, Lukáš MAIER, Stanislav STANDARA, Marek NEČAS, Filip LEMIERE a Radek MAREK. NMR study of covalent bonding of nitrogen-containing heterocyclic bases to quaternary protoberberine alkaloids. In PSE Young Sciencists` Meeting: Future Trends in Phytochemistry: Compounds-Enzymes-Genes. Germany, 2008, s. 14.
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Zobrazeno: 19. 9. 2024 06:57