Filtrování

    2025

    1. ŠIMURDOVÁ, Michaela; Tomáš STRHÁRSKY; Jiří KOS; Tomáš GONĚC; Alois ČÍŽEK a Josef JAMPÍLEK. Halogenated Cinnamanilides and Their Activity Against Selected Gram-Negative Bacteria. Online. In Halogenated Cinnamanilides and Their Activity against Selected Gram-negative Bacteria. ECSOC-29: MDPI, 2025, s. 1-7. ISSN 2673-4583. Dostupné z: https://doi.org/10.3390/ecsoc-29-26718.
    2. VRABLOVA, Lucia; Tomáš GONĚC; Petra MAJEROVA; Andrej KOVAC; Dominika KOS; Peter KOLLÁR; Jiří KOS; Alois CIZEK; Tereza KAUEROVÁ a Josef JAMPILEK. Insight into antistaphylococcal effect of chlorinated 1-hydroxynaphthalene-2-carboxanilides. ADMET AND DMPK. CROATIA: IAPC PUBLISHING, 2025, roč. 2025, č. 2684, s. 1-17. ISSN 1848-7718. Dostupné z: https://doi.org/10.5599/admet.2684.
    3. GONĚC, Tomáš; Jiří KOS; Dominika KOS; Michaela ŠIMURDOVÁ; Alois ČÍŽEK a Josef JAMPÍLEK. SEARCHING FOR EFFECTIVE ANTIMICROBIALS: PHENYLCARBAMOYLNAPHTHYL ALKYL CARBAMATES. In 53rd Conference Synthesis and Analysis of Drugs. 2025. ISBN 978-80-280-0773-7.
    4. KOS, Jiří; Tomáš STRHÁRSKY; Rodrigo TOSSO; Lucas GUTIERREZ; Dominika KOS; Jan JUŘICA; Ondřej ZENDULKA; Ondřej PEŠ; Jana GREGOROVÁ; Gilles DEGOTTE; Tomáš GONĚC; Michal ORAVEC; Veronika VOJACKOVA; Vladimir KRYSTOF; Alois ČÍŽEK; Pierre FRANCOTTE; Michel FREDERICH; Josef JAMPÍLEK a Daniel ENRIZ. Trifluoromethylcinnamanilides - Effective dual inhibitors of Mycobacterium smegmatis and Plasmodium falciparum. Bioorganic Chemistry. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE, 2025, roč. 154, January 2025, s. 1-22. ISSN 0045-2068. Dostupné z: https://doi.org/10.1016/j.bioorg.2024.107957.
    5. KOS, Jiří; Denis PAVELEK; Massoud KAYKHAII; Mark OLSEN; Josef JAMPÍLEK a Radoslav HALKO. Unveiling the transformative power of near-infrared spectroscopy in biomedical and pharmaceutical analysis: Trends, advancements, and applications. European Journal of Pharmaceutical Sciences. AMSTERDAM: ELSEVIER, 2025, roč. 212, September 2025, s. 1-20. ISSN 0928-0987. Dostupné z: https://doi.org/10.1016/j.ejps.2025.107175.

    2024

    1. PINDJAKOVA, Dominika; Sarka MASCARETTI; Jana HRICOVINIOVA; Jan HOSEK; Jana GREGOROVÁ; Jiří KOS; Alois CIZEK; Zuzana HRICOVINIOVA a Josef JAMPILEK. Critical view on antimicrobial, antibiofilm and cytotoxic activities of quinazolin-4(3H)-one derived schiff bases and their Cu(II) complexes. Heliyon. OXFORD: ELSEVIER, 2024, roč. 10, č. 7, s. 1-10. ISSN 2405-8440. Dostupné z: https://doi.org/10.1016/j.heliyon.2024.e29051.
    2. JAMPÍLEK, Jsoef; Tomáš STRHÁRSKY; Lucia VRÁBLOVÁ; Dominika KOS; Tomáš GONĚC a Jiří KOS. Design and Properties of New Multi-target Michael Acceptors. In Novel Trends in Chemistry, Research and Education 2024. 2024. ISBN 978-80-574-0370-8. Dostupné z: https://doi.org/10.33542/NTI-0370-8.
    3. Editorial of Special Issue "Current Trends in Chemistry Towards Biology" j - Publikace v odborném periodiku – kromě recenzovaných typů article, review a letter
      KOS, Jiří a Josef JAMPÍLEK. Editorial of Special Issue "Current Trends in Chemistry Towards Biology". International Journal of Molecular Sciences. BASEL: Molecular Diversity Preservation International, 2024, roč. 25, č. 13, s. 1-4. ISSN 1661-6596. Dostupné z: https://doi.org/10.3390/ijms25137307.
    4. JAMPÍLEK, Josef; Lucia VRÁBĽOVÁ; Dominika KOS; Tomáš GONĚC; Jiří KOS; Aleš IMRAMOVSKÝ a Alois ČÍŽEK. Effective Antimicrobial Agents Based on Ring-Substituted Hydroxyarylcarboxylic Acids. In The 20th Annual Congress of International Drug Discovery Science and Technology (IDDST-2024). 2024.

    2023

    1. STRHÁRSKY, Tomáš; Dominika PINDJAKOVÁ; Jaroslava JAMRICHOVÁ; Juliana LAVIČKOVÁ; Veronika KADLECOVÁ; Jiří KOS; Tomáš GONĚC a Josef JAMPÍLEK. Syntéza amidů kyseliny skořicové s antimikrobiální aktivitou. In 75. Zjazd chemikov. 2023. ISSN 1336-7242.
    2. SYNTHESIS OF ANTIBACTERIAL CINNAMAMIDES a - Konferenční abstrakt
      STRHÁRSKY, Tomáš; Dominika PINDJAKOVÁ; Jaroslava JAMRICHOVÁ; Juliana LAVIČKOVÁ; Veronika KADLECOVÁ; Kateřina KLEINEROVÁ; Jiří KOS; Tomáš GONĚC a Josef JAMPÍLEK. SYNTHESIS OF ANTIBACTERIAL CINNAMAMIDES. In 51st Conference Synthesis and Analysis of Drugs. 2023.
    3. BAK, Andrzej; Jiří KOS; Gilles DEGOTTE; Aleksandra SWIETLICKA; Tomáš STRHÁRSKY; Dominika PINDJAKOVA; Tomáš GONĚC; Adam SMOLINSKI; Pierre FRANCOTTE; Michel FREDERICH; Violetta KOZIK a Josef JAMPÍLEK. Towards Arginase Inhibition: Hybrid SAR Protocol for Property Mapping of Chlorinated N-arylcinnamamides. International Journal of Molecular Sciences. BASEL: MDPI, 2023, roč. 24, č. 4, s. 1-23. ISSN 1661-6596. Dostupné z: https://doi.org/10.3390/ijms24043611.

    2022

    1. KOS, Jiří; Gilles DEGOTTE; Dominika PINDJAKOVA; Tomáš STRHÁRSKY; Timotej JANKECH; Tomáš GONĚC; Pierre FRANCOTTE; Michel FREDERICH a Josef JAMPILEK. Insights into Antimalarial Activity of N-Phenyl-Substituted Cinnamanilides. Molecules. Basel: MDPI, 2022, roč. 27, č. 22, s. 1-10. ISSN 1420-3049. Dostupné z: https://doi.org/10.3390/molecules27227799.
    2. JAMPÍLEK, Josef; Jiří KOS; Tomáš STRHÁRSKY; Dominika PINDJAKOVÁ; Lucia VRÁBLOVÁ; Timotej JANKECH; Tomáš GONĚC a Alois ČÍŽEK. Investigation of Novel Halogenated Cinnamanilides. In The 11th International Conference on Biomedical Engineering and Biotechnology (ICBEB 2022). 2022.
    3. JAMPÍLEK, Josef; Dominika PINDJAKOVÁ; Tomáš GONĚC; Jiří KOS; Aleš IMRAMOVSKÝ a Alois ČÍŽEK. INVESTIGATIONS OF NEW DERIVATIVES OF β-HYDROXYARYLCARBOXYLIC ACIDS. In 12TH JMMC – JOINT MEETING ON MEDICINAL CHEMISTRY. 2022. ISBN 978-80-969474-9-2.
    4. STRHARSKY, Tomas; Dominika PINDJAKOVA; Jiří KOS; Lucia VRABLOVA; Hana MICHNOVA; Jan HOSEK; Nicol STRAKOVA; Veronika LELAKOVA; Lenka LEVA; Lenka KAVANOVA; Michal ORAVEC; Alois CIZEK a Josef JAMPILEK. Study of Biological Activities and ADMET-Related Properties of Novel Chlorinated N-arylcinnamamides. International Journal of Molecular Sciences. Basel: MDPI, 2022, roč. 23, č. 6, s. 1-20. ISSN 1422-0067. Dostupné z: https://doi.org/10.3390/ijms23063159.
    5. VRÁBLOVÁ, Lucia; Dominika PINDJAKOVÁ; Tomáš STRHÁRSKY; Tomáš GONĚC; Jiří KOS a Josef JAMPÍLEK. Štúdium interakcií orto-substituovaných anilidov 2- / 3- / 4-trifluórmetylškoricových kyselín. In XV. Medzinárodná konferencia Súčasný stav a perspektívy analytickej chémie v praxi. 2022. ISBN 978-80-227-5206-0.
    6. STRHÁRSKY, Tomáš; Dominika PINDJAKOVA; Jiří KOS; Lucia VRABLOVA; Pavel ŠMAK; Hana MICHNOVA; Tomáš GONĚC; Jan HOŠEK; Michal ORAVEC; Izabela JENDRZEJEWSKA; Alois ČÍŽEK a Josef JAMPILEK. Trifluoromethylcinnamanilide Michael Acceptors for Treatment of Resistant Bacterial Infections. International Journal of Molecular Sciences. Basel: Multidisciplinary Digital Publishing Institute, 2022, roč. 23, č. 23, s. 1-22. ISSN 1422-0067. Dostupné z: https://doi.org/10.3390/ijms232315090.

    2021

    1. PINDJAKOVÁ, Dominika; Lucia VRÁBLOVÁ; Tomáš STRHÁRSKY; Jiří KOS a Josef JAMPÍLEK. Investigation of interactions of ortho- and para-N-aryl-substituted 2-trifluoromethylcinnamanilides. In The 25th International Electronic Conference on Synthetic Organic Chemistry. 2021. Dostupné z: https://doi.org/10.3390/ecsoc-25-11651.
    2. KOS, Jiří; Tomáš GONĚC; Michal ORAVEC; Izabela JENDRZEJEWSKA a Josef JAMPÍLEK. Photosynthesis-Inhibiting Activity of N-(Disubstituted-phenyl)-3-hydroxynaphthalene-2-carboxamides. Molecules. MDPI Basel, 2021, roč. 26, č. 14, s. 1-9. ISSN 1420-3049. Dostupné z: https://doi.org/10.3390/molecules26144336.
    3. GAJDAR, Július; Jiří KOS; Tomáš GONĚC; Marie BRÁZDOVÁ; Zuzana SOLDÁNOVÁ; Miroslav FOJTA; Josef JAMPÍLEK; Jiří BAREK a Jan FISCHER. Substituent effect of ring-substituted 3-hydroxynaphthalene-2-carboxanilides and 2-hydroxynaphthalene-1-carboxanilides in relation to their electrochemical and biological activity. Journal of Electroanalytical Chemistry. Lausanne: Elsevier, 2021, roč. 899, October 2021, s. 1-8. ISSN 1572-6657. Dostupné z: https://doi.org/10.1016/j.jelechem.2021.115667.
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