Filtrování

    2025

    1. FARSA, Oldřich a Tomáš UHER. Aminopeptidase N: a multifunctional and promising target in medicinal chemistry. RSC ADVANCES. CAMBRIDGE: ROYAL SOC CHEMISTRY, 2025, roč. 15, č. 32, s. 26455-26472. ISSN 2046-2069. Dostupné z: https://doi.org/10.1039/d5ra03038b.
    2. ZIDEKOVA, Nela; Kristian PRSO; Marek PRSO; Milos JESENAK; Oldřich FARSA a Martin KERTYS. Development and Validation of a Rapid and Simple UHPLC-MS/MS Method for the Determination of Colchicine in Human Plasma. BIOMEDICAL CHROMATOGRAPHY. HOBOKEN: WILEY, 2025, roč. 39, č. 11, s. 1-9. ISSN 0269-3879. Dostupné z: https://doi.org/10.1002/bmc.70222.
    3. MURGAŠOVÁ, Veronika; Jovana LISIČIĆ; Ondřej SMIŠTÍK; Jan HOŠEK a Oldřich FARSA. SYNTHESIS AND BIOLOGICAL EVALUATION OF BASIC AMINOACETOPHENONE-DERIVED KETIMINES. In 59th Advances in Organic, Bioorganic and Pharmaceutical Chemistry: "Liblice 2025". 2025.
    4. MURGAŠOVÁ, Veronika a Oldřich FARSA. SYNTHESIS AND EVALUATION OF AMINOACETOPHENONE-DERIVED KETIMINES AS POTENTIAL THERAPEUTIC AGENTS. In 53rd Conference Synthesis and Analysis of Drugs 2025. 2025. ISBN 978-80-280-0773-7.
    5. FARSA, Oldřich. Synthesis of valproic acid for medicinal chemistry practical classes. CHEMISTRY TEACHER INTERNATIONAL. BERLIN: WALTER DE GRUYTER GMBH, 2025, roč. 7, č. 3, s. 563-573. ISSN 2569-3263. Dostupné z: https://doi.org/10.1515/cti-2025-0028.

    2023

    1. Aminopeptidase N as a potential drug target J - Článek v odborném periodiku
      FARSA, Oldřich; Veronika BALLAYOVÁ; Radka ŽÁČKOVÁ a Peter ZUBÁČ. Aminopeptidase N as a potential drug target. European Pharmaceutical Journal. Sciendo, 2023, roč. 70, s2, s. „AoP,1“-„2“, 2 s. ISSN 2453-6725. Dostupné z: https://doi.org/10.2478/afpuc-2024-0002.
    2. FARSA, Oldřich; Veronika BALLAYOVÁ; Radka ŽÁČKOVÁ a Peter ZUBÁČ. Aminopeptidase N as a potential drug target. In Ladislav Habala. 51st Conference Synthesis and Analsis of Drugs, Book of Abstracts. 1st ed. Bratislava: Faculty of Pharmacy, Comenius University in Bratislava, 2023, s. 13-13, 55 s. ISBN 978-80-280-0324-1.
    3. SCHIFF BASES AS POTENTIAL THERAPEUTIC AGENTS k - Prezentace na konferencích
      BALLAYOVÁ, Veronika; Tereza KAUEROVÁ; Peter KOLLÁR a Oldřich FARSA. SCHIFF BASES AS POTENTIAL THERAPEUTIC AGENTS. In Student Scientific Conference MUNI Pharm. Doctoral Students 2023. 2023. ISBN 978-80-280-0324-1.
    4. BALLAYOVÁ, Veronika; Tereza KAUEROVÁ; Peter KOLLÁR a Oldřich FARSA. SCHIFF BASES AS POTENTIAL THERAPEUTIC AND ANTICANCER AGENTS. In 51st Conference Synthesis and Analysis of Drugs, 2023. 2023. Dostupné z: https://doi.org/10.2478/afpuc-2023-0022.

    2022

    1. FARSA, Oldřich; Veronika BALLAYOVÁ; Radka ŽÁČKOVÁ; Peter KOLLÁR; Tereza KAUEROVÁ a Peter ZUBÁČ. Aminopeptidase N Inhibitors as Pointers for Overcoming Antitumor Treatment Resistance. International Journal of Molecular Sciences. Basel: Multidisciplinary Digital Publishing Institute, 2022, roč. 23, č. 17, s. 1-15. ISSN 1422-0067. Dostupné z: https://doi.org/10.3390/ijms23179813.
    2. FARSA, Oldřich; Veronika BALLAYOVÁ; Radka ŽÁČKOVÁ; Peter KOLLÁR; Tereza KAUEROVÁ a Peter ZUBÁČ. Aromatic Schiff bases as aminopeptidase N inhibitors. In 50th conference Syntesis and Analysis of Drugs. 2022. ISBN 978-80-280-0110-0.
    3. BALLAYOVÁ, Veronika; Radka ŽÁČKOVÁ a Oldřich FARSA. DETERMINATION OF INHIBITORY ACTIVITY OF AMINOPEPTIDASE N BY USING HIGH-PERFORMANCE LIQUID CHROMATOGRAPHY. 2022. ISBN 978-80-280-0105-6.
    4. BALLAYOVÁ, Veronika; Radka ŽÁČKOVÁ; Tereza KAUEROVÁ; Peter KOLLÁR a Oldřich FARSA. SCHIFF BASES AS POTENTIAL INHIBITORS OF AMINOPEPTIDASE N AS ANTICANCER AGENTS. 2022.

    2021

    1. BALLAYOVÁ, Veronika; Peter ZUBÁČ; Radka ŽÁČKOVÁ a Oldřich FARSA. Basic derivatives of aromatic-aliphatic ketones as potential inhibitors of aminopeptidase N. In Student scientific conference MUNI PHARM 2021. 2021. ISBN 978-80-210-9870-1.
    2. ZUBÁČ, Peter a Oldřich FARSA. DESIGN, SYNTHESIS AND STRUCTURE-BASED OPTIMIZATION OF POTENTIAL PHENOTHIAZINE ANTIMICROBIALS. In 49th Conference Synthesis and Analysis of Drugs 2021 Hradec Králové. 2021.
    3. ŽÁČKOVÁ, Radka; Veronika BALLAYOVÁ; Peter ZUBÁČ a Oldřich FARSA. Determination of aminopeptidase N inhibitory activity of newly synthesised nitrogenous compounds. In Student Scientific Conference Muni Pharm 2021. 2021. ISBN 978-80-210-9870-1.
    4. FARSA, Oldřich a Peter ZUBÁČ. Protein and Small-Molecule Leucopoiesis and Thrombopoiesis Stimulators. Mini-reviews in medicinal chemistry. Sharjah: Betham Science Publ Ltd., 2021, roč. 21, č. 13, s. 1638-1645. ISSN 1389-5575. Dostupné z: https://doi.org/10.2174/1389557521999201230195926.
    5. BALLAYOVÁ, Veronika; Peter ZUBÁČ; Radka ŽÁČKOVÁ a Oldřich FARSA. Synthesis of Schiff bases with potential therapeutic activity. In 49th Conference Synthesis and Analysis of Drugs. 2021.

    2020

    1. PADRTOVÁ, Tereza; Pavlína MARVANOVÁ; Renata KUBÍNOVÁ; Jozef CSÖLLEI; Oldřich FARSA; Tomáš GONĚC; Klára ODEHNALOVÁ; Radka OPATŘILOVÁ; Jiří PAZOUREK; Alice SYCHROVÁ; Karel ŠMEJKAL a Petr MOKRÝ. Indol-2-Carboxylic Acid Esters Containing N-Phenylpiperazine Moiety - Preparation and Cholinesterase-inhibiting Activity. Current organic synthesis. Sharjah: Bentham Science Publ Ltd, 2020, roč. 17, č. 7, s. 576-587. ISSN 1570-1794. Dostupné z: https://doi.org/10.2174/1570179417666200619132218.

    2019

    1. FARSA, Oldřich a Peter ZUBÁČ. Erythropoetins in Therapy from the Point of View of a Medicinal Chemist. CHEMICKÉ LISTY. Praha: Česká společnost chemická, 2019, roč. 113, č. 9, s. 540-544. ISSN 0009-2770.

    2018

    1. FARSA, Oldřich a Peter ZUBÁČ. Hematopoiteic factors are not only proteins. In Optařilová R., Marvanová P. Book of Abstracts SAL 2018 Brno. Brno: Veterinární a farmaceutická univerzita Brno, 2018, s. 26-26. ISBN 978-80-7305-806-7.
    2. VYSLOUŽIL, Jakub; David VETCHÝ; Jiří ZEMAN; Oldřich FARSA; Aleš FRANC; Jan GAJDZIOK; Jan VYSLOUŽIL; Katarina FICERIOVA; Pavel KULICH; Zbynek KOBLIHA a Vladimir PITSCHMANN. Pellet patented technology for fast and distinct visual detection of cholinesterase inhibitors in liquids. Journal of Pharmaceutical and Biomedical Analysis. Amsterdam: Elsevier Science BV, 2018, roč. 161, August, s. 206-213. ISSN 0731-7085. Dostupné z: https://doi.org/10.1016/j.jpba.2018.08.050.

    2017

    1. FARSA, Oldřich; Jakub KÁŇA; Irena MACKŮ; Jana ŽELAZKOVÁ; Jana PODLIPNÁ; Aleš CIRKVA; Jaroslav MAXA a Kamil ŠŤASTNÝ. SYNTHESIS AND AMINOPEPTIDASE N INHIBITING ACTIVITY OF 3-(NITROPHENOXYMETHYL)-[1,3,2]DIOXABOROLAN-2-OLS AND THEIR OPEN ANALOGUES. ACTA POLONIAE PHARMACEUTICA. WARSAW: POLSKIE TOWARZYSTWO FARMACEUTYCZNE, 2017, roč. 74, č. 1, s. 127-135. ISSN 0001-6837.

    2016

    1. FARSA, Oldřich a Matěj HALUSKA. A SINGLE- AND MULTIPARAMETRIC QSAR STUDY OF AMINOPEPTIDASE N INHIBITORS. FARMACIA. BUCURESTI: SOC STIINTE FARMACEUTICE ROMANIA, 2016, roč. 64, č. 2, s. 283-290. ISSN 0014-8237.
    2. FARSA, Oldřich. Molární substituce substituovaných oligo- a polysacharidů NMR. Online. In Doležal M. 45. konference SYNTÉZA A ANALÝZA LÉČIV. Sborník. Hradec Králové: Česká farmaceutická společnost ČLS JEP, 2016, s. S-9, 2 s.

    2015

    1. FARSA, Oldřich. Aminopeptidase N inhibition could be involved in the anti-angiogenic effect of dobesilates. Journal of the Serbian Chemical Society. 2015. Dostupné z: https://doi.org/10.2298/JSC131128032F.
    2. FARSA, Oldřich. From an old drug to a new one: synthesis of valproate from 5,​5-​dipropylbarbituric acid. 2015.

    2014

    1. KUBÍNOVÁ, Renata; R. PORIZKOVA; Alice SYCHROVÁ; Oldřich FARSA; Zuzana HANÁKOVÁ; A. BACINSKA; Alois ČÍŽEK a Marie VALENTOVÁ. Antimicrobial and enzyme inhibitory activities of the constituents of Plectranthus madagascariensis (Pers.) Benth. Journal of Enzyme Inhibition and Medicinal Chemistry. UK: Taylor & Francis, 2014, roč. 29, č. 5, s. 749-752. ISSN 1475-6366. Dostupné z: https://doi.org/10.3109/14756366.2013.848204.

    2003

    1. PAZOURKOVÁ, M; Antonín LOJEK; Milan ČÍŽ; Lukáš KUBALA; L BENEŠ a Oldřich FARSA. Antioxidative activity of pyridoindoles and N-(alkoxyphenyl)-2-(2-oxo-1-aza-1-cykloalkyl)acetamines in biological, enzymatic a chemical systems. Čes. Slov. Fram. 2003, roč. 52, č. 4, s. 171-175. ISSN 1210-7816.
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